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HAART Chart - Approved Antiretroviral Drugs

From the Winter 2007 edition of the Bulletin of Experimental Treatments for AIDS
Generic (Common) Name Brand Name Company Year Approved
Protease Inhibitors (PIs)
amprenavir Agenerase GlaxoSmithKline 1999; discontinued 2004
atazanavir Reyataz Bristol-Myers Squibb 2003
darunavir (TMC114) Prezista Tibotec 2006
fosamprenavir Lexiva (U.S.); Telzir (Europe) GlaxoSmithKline 2003
indinavir Crixivan Merck 1996
lopinavir/ritonavir Kaletra Abbott 2000; Meltrex formulation 2005
nelfinavir Viracept Pfizer 1997
ritonavir Norvir Abbott 1996
saquinavir Invirase (hard-gel)
Fortovase (soft-gel)
Roche 1995
1997; withdrawn 2005
tipranavir Aptivus Boehringer Ingelheim 2005
Nucleoside/Nucleotide Reverse Transcriptase Inhibitors (NRTIs)
abacavir Ziagen GlaxoSmithKline 1998
didanosine (ddI) Videx Bristol-Myers Squibb 1989; extended release Videx EC 2000
emtricitabine (FTC) Emtriva Gilead 2003
lamivudine (3TC) Epivir GlaxoSmithKline 1995
stavudine (d4T) Zerit Bristol-Myers Squibb 1994
tenofovir DF Viread Gilead 2002
zalcitabine (ddC) Hivid Roche 1992; withdrawn 2005
zidovudine (AZT) Retrovir GlaxoSmithKline 1987
Non-Nucleoside Reverse Transcriptase Inhibitors (NNRTIs)
delavirdine Rescriptor Pfizer 1997
efavirenz Sustiva (U.S.); Stocrin (elsewhere) Bristol-Myers Squibb 1998
nevirapine Viramune Boehringer Ingelheim 1996
Entry/Fusion Inhibitors
enfuvirtide (T-20) Fuzeon Trimeris 2003
Fixed-Dose Combinations
lamivudine/abacavir (NRTI) Epzicom (U.S.); Kivexa (Europe) GlaxoSmithKline 2004
tenofovir/emtricitabine (NRTI) Truvada Gilead 2004
tenofovir/emtricitabine/
efavirenz (NRTI/NNRTI)
Atripla Gilead/Bristol-Myers Squibb 2006
zidovudine/lamivudine (NRTI) Combivir GlaxoSmithKline 1997
zidovudine/lamivudine/abacavir (NRTI) Trizivir GlaxoSmithKline 2000
Page last updated: 1/1/2007


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